Studies towards the synthesis of indolizin-5(3H)-one derivatives and related 6,5-azabicyclic scaffolds by ring-closing metathesis
MS Frei, MK Bilyard, TA Alanine, WRJD Galloway, JE Stokes, DR Spring
– Bioorganic and Medicinal Chemistry
(2015)
23,
2666
(DOI: 10.1016/j.bmc.2014.11.037)
Divergent and concise total syntheses of dihydrochalcones and 5-deoxyflavones recently isolated from Tacca species and Mimosa diplotricha
TH Sum, TJ Sum, JE Stokes, WRJD Galloway, DR Spring
– Tetrahedron
(2015)
71,
4557
(DOI: 10.1016/j.tet.2015.02.017)
The Pseudomonas Quinolone Signal (PQS)
T Sams, Y Baker, J Hodgkinson, J Gross, D Spring, M Welch
– Israel Journal of Chemistry
(2015)
56,
282
(DOI: 10.1002/ijch.201400128)
Enantioselective Synthesis of Chromanones via a Peptidic Phosphane Catalyzed Rauhut-Currier Reaction
RJH Scanes, O Grossmann, A Grossmann, DR Spring
– Organic Letters
(2015)
17,
2462
(DOI: 10.1021/acs.orglett.5b00971)
A two-component 'double-click' approach to peptide stapling.
YH Lau, Y Wu, P de Andrade, WRJD Galloway, DR Spring
– Nature Protocols
(2015)
10,
585
(DOI: 10.1038/nprot.2015.033)
Divergent and concise total syntheses of dihydrochalcones and 5-deoxyflavones recently isolated from <i>Tacca</i> species and <i>Mimosa diplotricha</i>
TH Sum, TJ Sum, JE Stokes, WRJD Galloway, DR Spring
– Tetrahedron
(2015)
71,
4557
(DOI: 10.1016/j.tet.2015.02.017)
Diversity oriented synthesis of macrocycles using a build/couple/pair/diversity strategy
F Nie, D Kunciw, J Stokes, D Spring
– ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
(2015)
250,
A diversity-oriented synthesis strategy enabling the combinatorial-type variation of macrocyclic peptidomimetic scaffolds.
A Isidro-Llobet, K Hadje Georgiou, WRJD Galloway, E Giacomini, MR Hansen, G Méndez-Abt, YS Tan, L Carro, HF Sore, DR Spring
– Organic & Biomolecular Chemistry
(2015)
13,
4570
(DOI: 10.1039/c5ob00371g)
Using small molecules to solve big problems
J Stokes, D Spring
– ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
(2015)
250,
Studies towards the synthesis of indolizin-5(3H)-one derivatives and related 6,5-azabicyclic scaffolds by ring-closing metathesis.
MS Frei, MK Bilyard, TA Alanine, WRJD Galloway, JE Stokes, DR Spring
– Bioorganic & Medicinal Chemistry
(2014)
23,
2666
(DOI: 10.1016/j.bmc.2014.11.037)
Multifunctional supramolecular polymer networks as next-generation consolidants for archaeological wood conservation.
Z Walsh, E-R Janeček, JT Hodgkinson, J Sedlmair, A Koutsioubas, DR Spring, M Welch, CJ Hirschmugl, C Toprakcioglu, JR Nitschke, M Jones, OA Scherman
– Proceedings of the National Academy of Sciences
(2014)
111,
17743
(DOI: 10.1073/pnas.1406037111)
Linear Aliphatic Dialkynes as Alternative Linkers for Double-Click Stapling of p53-Derived Peptides
YH Lau, P de Andrade, GJ McKenzie, AR Venkitaraman, DR Spring
– Chembiochem
(2014)
15,
2680
(DOI: 10.1002/cbic.201402374)
Diversity‐Oriented Synthesis: Developing New Chemical Tools to Probe and Modulate Biological Systems
WRJD Galloway, D Wilcke, F Nie, K Hadje-Georgiou, L Laraia, DR Spring
(2014)
9783527336111,
379
(DOI: 10.1002/9783527687503.ch26)
Diversity‐Oriented Synthesis of Drug‐Like Macrocyclic Scaffolds Using an Orthogonal Organo‐ and Metal Catalysis Strategy
A Grossmann, S Bartlett, M Janecek, JT Hodgkinson, DR Spring
– Angewandte Chemie (International ed. in English)
(2014)
53,
13093
(DOI: 10.1002/anie.201406865)
Synthesis of a novel polycyclic ring scaffold with antimitotic properties
E Alza, L Laraia, BM Ibbeson, S Collins, WRJD Galloway, JE Stokes, AR Venkitaraman, DR Spring
– Chemical Science
(2014)
6,
390
(DOI: 10.1039/c4sc02547d)
Peptide stapling techniques based on different macrocyclisation chemistries.
YH Lau, P de Andrade, Y Wu, DR Spring
– Chemical Society Reviews
(2014)
44,
91
(DOI: 10.1039/c4cs00246f)
Concise synthesis of substituted quinolizin-4-ones by ring-closing metathesis
TA Alanine, WRJD Galloway, TM McGuire, DR Spring
– European Journal of Organic Chemistry
(2014)
2014,
5767
(DOI: 10.1002/ejoc.201402648)
Concise Synthesis of Substituted Quinolizin‐4‐ones by Ring‐Closing Metathesis
TA Alanine, WRJD Galloway, TM Mcguire, DR Spring
– European Journal of Organic Chemistry
(2014)
2014,
5767
(DOI: 10.1002/ejoc.201402648)
Toxicity of six plant extracts and two pyridone alkaloids from Ricinus communis against the malaria vector Anopheles gambiae.
SW Wachira, S Omar, JW Jacob, M Wahome, HT Alborn, DR Spring, DK Masiga, B Torto
– Parasites & Vectors
(2014)
7,
312
(DOI: 10.1186/1756-3305-7-312)
Arene C–H functionalisation using a removable/modifiable or a traceless directing group strategy
F Zhang, DR Spring
– Chem. Soc. Rev.
(2014)
43,
6906
(DOI: 10.1039/c4cs00137k)