Research Associate
Publications
Targeted covalent inhibitors of MDM2 using electrophile-bearing stapled peptides
– Chemical communications (Cambridge, England)
(2019)
55,
7914
(doi: 10.1039/c9cc04022f)
Efficient development of stable and highly functionalised peptides targeting the CK2α/CK2β protein-protein interaction.
– Chem Sci
(2019)
10,
5056
(doi: 10.1039/c9sc00798a)
Two-component stapling of biologically active and conformationally constrained peptides: past, present and future
– Advanced Therapeutics
(2018)
1,
1800052
(doi: 10.1002/adtp.201800052)
Novel non-ATP competitive small molecules targeting the CK2 α/β interface
– Bioorganic & Medicinal Chemistry
(2018)
26,
3016
(doi: 10.1016/j.bmc.2018.05.011)
Stapled peptides as a new technology to investigate protein–protein interactions in human platelets
– Chemical science
(2018)
9,
4638
(doi: 10.1039/x0xx00000x)
Second-generation CK2α inhibitors targeting the αD pocket.
– Chemical science
(2018)
9,
3041
(doi: 10.1039/c7sc05122k)
A fragment-based approach leading to the discovery of a novel binding site and the selective CK2 inhibitor CAM4066.
– Bioorganic and Medicinal Chemistry
(2017)
25,
3471
(doi: 10.1016/j.bmc.2017.04.037)
Binding Mode and Induced Fit Predictions for Prospective Computational Drug Design.
– Journal of Chemical Information and Modeling
(2016)
56,
774
(doi: 10.1021/acs.jcim.5b00744)
Database Extraction of Metabolite Information of Drug Candidates: Analysis of 27 AstraZeneca Compounds with Human Absorption, Distribution, Metabolism, and Excretion Data
– Drug metabolism and disposition: the biological fate of chemicals
(2016)
44,
732
(doi: 10.1124/dmd.115.067850)
Salicylketoximes That Target Glucose Transporter 1 Restrict Energy Supply to Lung Cancer Cells
– ChemMedChem
(2015)
10,
1892
(doi: 10.1002/cmdc.201500320)
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