
Principle Research Associate
Publications
Structure Based Discovery of Inhibitors of CYP125 and CYP142 from Mycobacterium tuberculosis.
– Chemistry
(2023)
e202203868
(DOI: 10.1002/chem.202203868)
Chemical Validation of Mycobacterium tuberculosis Phosphopantetheine Adenylyltransferase Using Fragment Linking and CRISPR Interference
– Angewandte Chemie
(2023)
(DOI: 10.1002/ange.202300221)
Chemical Validation of Mycobacterium tuberculosis Phosphopantetheine Adenylyltransferase Using Fragment Linking and CRISPR Interference
– Angewandte Chemie International Edition
(2023)
(DOI: 10.1002/anie.202300221)
Microfluidic preparation of composite hydrogel microparticles for the staining of microalgal cells.
– Colloids Surf B Biointerfaces
(2022)
221,
113026
Development of potent inhibitors by fragment‐linking strategies
– Chem Biol Drug Des
(2022)
100,
469
(DOI: 10.1111/cbdd.14120)
Structural Characterization of Mycobacterium abscessus Phosphopantetheine Adenylyl Transferase Ligand Interactions: Implications for Fragment-Based Drug Design
– Front Mol Biosci
(2022)
9,
880432
(DOI: 10.3389/fmolb.2022.880432)
Potential therapeutic targets from Mycobacterium abscessus ( Mab ): recently reported efforts towards the discovery of novel antibacterial agents to treat Mab infections
– RSC medicinal chemistry
(2022)
13,
392
(DOI: 10.1039/d1md00359c)
Discovery of Novel Inhibitors of Uridine Diphosphate-N-Acetylenolpyruvylglucosamine Reductase (MurB) from Pseudomonas aeruginosa, an Opportunistic Infectious Agent Causing Death in Cystic Fibrosis Patients.
– J Med Chem
(2022)
65,
2149
(DOI: 10.1021/acs.jmedchem.1c01684)
Development of Inhibitors of SAICAR Synthetase (PurC) from Mycobacterium abscessus Using a Fragment-Based Approach.
– ACS Infect Dis
(2022)
8,
296
(DOI: 10.1021/acsinfecdis.1c00432)
A new strategy for hit generation: Novel in cellulo active inhibitors of CYP121A1 from Mycobacterium tuberculosis via a combined X-ray crystallographic and phenotypic screening approach (XP screen)
– Eur J Med Chem
(2022)
230,
114105
(DOI: 10.1016/j.ejmech.2022.114105)
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