Publications
Using a Fragment-Based Approach to Identify Alternative Chemical Scaffolds Targeting Dihydrofolate Reductase from Mycobacterium tuberculosis.
– ACS Infect Dis
(2020)
6,
2192
(DOI: 10.1021/acsinfecdis.0c00263)
Fragment-based discovery of a new class of inhibitors targeting mycobacterial tRNA modification
– Nucleic Acids Res
(2020)
48,
8099
(DOI: 10.1093/nar/gkaa539)
Fragment-based design of mycobacterium tuberculosis inha inhibitors
– Journal of Medicinal Chemistry
(2020)
63,
4749
(DOI: 10.1021/acs.jmedchem.0c00007)
Covalent inactivation of Mycobacterium thermoresistibile inosine-5′-monophosphate dehydrogenase (IMPDH)
– Bioorganic & Medicinal Chemistry Letters
(2020)
30,
126792
(DOI: 10.1016/j.bmcl.2019.126792)
Allosteric Small-Molecule Serine/Threonine Kinase Inhibitors.
– Adv Exp Med Biol
(2019)
1163,
253
(DOI: 10.1007/978-981-13-8719-7_11)
Targeting of fumarate hydratase from Mycobacterium tuberculosis using allosteric inhibitors with a dimeric-binding mode
– J Med Chem
(2019)
62,
10586
(DOI: 10.1021/acs.jmedchem.9b01203)
Structural insights into Escherichia coli phosphopantothenoylcysteine synthetase by native ion mobility-mass spectrometry.
– Biochemical Journal
(2019)
476,
3125
(DOI: 10.1042/bcj20190318)
Development of inhibitors against mycobacterium abscessus tRNA (m1G37) Methyltransferase (TrmD) Using Fragment-Based Approaches
– Journal of medicinal chemistry
(2019)
62,
7210
(DOI: 10.1021/acs.jmedchem.9b00809)
Structure-guided Fragment-based Drug Discovery at the Synchrotron: Screening Binding Sites and Correlations with Hotspot Mapping
– Philosophical Transactions of the Royal Society A: Mathematical, Physical and Engineering Sciences
(2019)
377,
20180422
(DOI: 10.1098/rsta.2018.0422)
meta‐Nitration of Arenes Bearing ortho/para Directing Group(s) Using C−H Borylation
– Chemistry - A European Journal
(2019)
25,
8018
(DOI: 10.1002/chem.201901633)
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